Listar por materia "Multicomponent reactions"
Mostrando publicaciones 1-3 de 3
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A peptide backbone stapling strategy enabled by the multicomponent incorporation of amide n-substituents
(2019)The multicomponent backbone N-modification of peptides on solid-phase is presented as a powerful and general method to enable peptide stapling at the backbone instead of the side chains. This work shows that a variety of ...
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Synthesis of lactam-bridged and lipidated cyclo-peptides as promising anti-phytopathogenic agents
(2020)Antimicrobial resistance to conventional antibiotics and the limited alternatives to combat plant-threatening pathogens are worldwide problems. Antibiotic lipopeptides exert remarkable membrane activity, which usually is ...
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Ugi reaction-derived prolyl peptide catalysts grafted on the renewable polymer polyfurfuryl alcohol for applications in heterogeneous enamine catalysis
(2019)The multicomponent synthesis of prolyl pseudo-peptide catalysts using the Ugi reaction with furfurylamines or isocyanides is described. The incorporation of such a polymerizable furan handle enabled the subsequent ...